20th Drug Discovery Chemistry

Drug Discovery Chemistry is a premier gathering for medicinal, biophysical, and computational chemists advancing small molecule and macrocyclic therapeutics. Featuring leaders from top pharma and biotech, the conference delivers cutting-edge insights on discovery and optimization challenges, with flexible tracks that let attendees tailor their experience across fragment-based discovery, targeted protein degradation, beyond-Rule-of-5 modalities, and more.

Held at the Hilton San Diego Bayfront, the event combines world-class science with high-impact networking, connecting researchers across industry and academia. Plenary keynotes from noted innovators spotlight practical strategies, emerging chemistries, and translational case studies—equipping teams to accelerate the path from concept to clinic.